Author ORCID Identifier

0000-0003-0390-7663

Date of Graduation

8-2024

Document Type

Dissertation (PhD)

Program Affiliation

Genetics and Epigenetics

Degree Name

Doctor of Philosophy (PhD)

Advisor/Committee Chair

Michael J. Galko

Committee Member

Mark Bedford

Committee Member

George Eisenhoffer

Committee Member

Honami Naora

Committee Member

Sheng Zhang

Abstract

Paclitaxel (PTX), a chemotherapeutic that alters microtubule dynamics, is known to induce nociceptive hypersensitivity and sensory neuron damage in human patients and in Drosophila larvae. We used a modified feeding protocol to establish a genetically tractable Drosophila model of PTX-induced hypersensitivity. Larvae fed PTX exhibited hypersensitivity to thermal and mechanical stimuli. Thermal hypersensitivity was observed at low concentrations of PTX (even below 1 μM per ml of food), begins within 8 hours of PTX feeding, and did not completely resolve at the larval stage. Live imaging of peripheral thermal nociceptors showed that this hypersensitivity precedes observable neuronal damage. At low concentrations, PTX caused hyper-sprouting of tertiary dendritic spines in peripheral nociceptors. At high concentrations, it caused dendritic degradation. We used this model of PTX-induced hypersensitivity to explore its molecular/genetic basis. Of particular interest was insulin-like signaling (ILS) which regulates the persistence of damage-induced hypersensitivity. RNAi targeting the insulin receptor (InR) in nociceptors increased PTX- induced hypersensitivity. However, insulin-like peptide 4 (ILP4), was only required for PTX- induced thermal hypersensitivity at 10 μM. In summary, our model of PTX-induced hypersensitivity revealed a disconnect between hypersensitivity and neuronal morphology and a genetic separation of ILP4 and InR in PTX-induced hypersensitivity.

Keywords

Drosophila, Paclitaxel, nociception, ILP4, nociceptive hypersensitivity

Available for download on Tuesday, February 11, 2025

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