Faculty, Staff and Student Publications

Language

English

Publication Date

12-24-2024

Journal

International Journal of Molecular Sciences

DOI

10.3390/ijms26010016

PMID

39795874

PMCID

PMC11720453

PubMedCentral® Posted Date

12-24-2024

PubMedCentral® Full Text Version

Post-print

Abstract

Pseudoachondroplasia (PSACH), a severe dwarfing condition characterized by impaired skeletal growth and early joint degeneration, results from mutations in cartilage oligomeric matrix protein (COMP). These mutations disrupt normal protein folding, leading to the accumulation of misfolded COMP in chondrocytes. The MT-COMP mouse is a murine model of PSACH that expresses D469del human COMP in response to doxycycline and replicates the PSACH chondrocyte and clinical pathology. The basis for the mutant-COMP pathology involves endoplasmic reticulum (ER) stress signaling through the PERK/eIF2α/CHOP pathway. C/EBP homologous protein (CHOP), in conjunction with a TNFα inflammatory process, upregulates mTORC1, hindering autophagy clearance of mutant COMP protein. Life-long joint pain/degeneration diminishes quality of life, and treatments other than joint replacements are urgently needed. To assess whether molecules that reduce CHOP activity should be considered as a potential treatment for PSACH, we evaluated MT-COMP mice with 50% CHOP (MT-COMP/CHOP

Keywords

Achondroplasia, Femur, Transcription Factor CHOP, Cartilage Oligomeric Matrix Protein, Mice, Transgenic, Arthralgia, Joint Diseases, Chondrocytes, Growth Plate, Cell Death, Mice, Inbred C57BL, Male, Animals, Mice, cartilage oligomeric matrix protein, COMP, autophagy, ASO, CHOP, chondrocyte, ER stress, joint degeneration

Published Open-Access

yes

Included in

Dentistry Commons

Share

COinS
 
 

To view the content in your browser, please download Adobe Reader or, alternately,
you may Download the file to your hard drive.

NOTE: The latest versions of Adobe Reader do not support viewing PDF files within Firefox on Mac OS and if you are using a modern (Intel) Mac, there is no official plugin for viewing PDF files within the browser window.